Melanotan IIbụ synthetic cyclic heptapeptide analọg nkeα-melanocyte na-akpali akpali hormone (α-MSH), tolitere kana-akpali melanogenesis, kwaliteNchekwa UV, ma gbanweemmekọahụ na metabolic ọrụ. Ọ na-eme dị ka aagonist anaghị ahọpụtanke melanocortin receptors, karịsịaMC1R, MC3R, naMC4R.
Na mbụ gụrụ maka yatanningnafotoprotectiveNjirimara, Melanotan II egosikwala mmetụta nankwalite libido, mkpochapụ agụụ, naike itule, na-eme ka ọ bụrụ peptide nyocha multifunctional nwere mmasị na dermatology, endocrinology, na ọgwụ mmekọahụ.
Melanotan II na-arụ ọrụ site na ịgbalite ọtụtụ ndị na-anabata melanocortin:
MC1R: Na-akpalimmepụta nke melanin→ na-abawanye pigmenti anụ ahụ na nchebe UV
MC3R / MC4R: Abanye nanjikwa agụụ, nkwalite libido, naike homeostasis
Na-agafe ihe mgbochi ụbụrụ ọbara, na-emetụta Central neurohormonal ụzọ
Ọ bụ ezie na akwadoghị maka iji ahụike, Melanotan II na-amụ nke ọma maka ihe ndị a:
Na-akwaliteeumelanin njikọ, na-eduga naeke tanning
Na-enyefoto-echebe mmetụtana-enweghị anwụ ikpughe
Enwere ike ibelata ihe ize ndụ cancer anụ ahụ n'ime ndị nwere akpụkpọ ahụ
Egosiri yamụbaa libido na agụụ mmekọahụma ndị nwoke ma ndị nwanyị
Agụrụ akwụkwọ dị ka ọgwụgwọ nwere ike maka yaỌkpụkpụ erectile (ED)site na MC4R ịgbalite
Meebelata agụụ na iri nrisite na ime ihe na ụzọ hypothalamic
Ihe mgbakwunye nwere ike ịbanyennyocha oke ibu
Ịdị ọcha dị elu ≥ 99%(HPLC & LC-MS kwadoro)
Synthesized siteNgwakọta peptide siri ike (SPPS)
Endotoxin dị ala, ihe mgbaze dị ala
Dị naR&D n'ọtụtụ azụmaahịa