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Deflazacot nwere mgbochi mkpali, mgbochi nfụkasị, ma na-abawanye mmetụta gloconeogenesis

Nkọwa mkpụmkpụ:

Na-agbaze na-emegharị: 255-256.5 Celsius C

Ntugharị ndị akọwapụtara: D + 62.3 Celsius (c = 05inchloroform)

Isi mmiri: 595.4 ± ± 50.0 Celsius C (buru amụma)

Nnọọ: 1.41

Ọnọdụ nchekwa: 2-8 Celsius C

Solubality: DMSO: ≥20MG / ml

Acidity Cofiefy: (Pka) 14.30 ± 0.70 (buru amụma)

Udi: ntụ

Agba: Black


Nkọwa nke ngwaahịa

Mkpado Ngwaahịa

Nkọwa nke ngwaahịa

Aha Deflazacort
Nọmba 14484-47-0
Molular C25H31NO6
Molular ibu 441.52
Nọmba einecs 238-483-7
Isi mmiri 595.4 ± 50.0 Celsius C
Nko 98%
Storaji Achịcha na okpomoku
Odidi Nzu otite
Agba Ucha
Mbukota Akpa Pear + Aluminom akpa

Myiri

16-D) Oxazole-Dione-3,20, 11-beta, 21-behacydroxy-h-Pretyloxy-H-Methyloxy-21'-methylox-1,5-tetradeh ydropropyoregnole [17,16-d]

Mmetụta ọgwụ

Ngosiputa
N'ihi na nke abụọ ma ọ bụ nke abụọ na-adịghị mma, ọrịa na-egbu egbu, ọrịa coldrometic, ọrịa hediopattic, na nfụkasị nke ọgwụ mgbochi maka ọgwụgwọ nke Fulmany ma na-ekesa ụkwara akwara.

Mkpachapụ anya
(1) Dị ka glucocortortoids ndị ọzọ, ọ na-eke contraindiation maka ọrịa na-efe efe.
(2) Jiri nlezianya na-akpachara anya na SendTerlinal Agrerynation na-adịbeghị anya, odida, odida, ọbara mgbali elu, ọrịa shuga, Myastenia gravis na ọrịa ndị ọzọ. Ime ka ụmụ nwanyị dị ime.

Mkpakọrịta ọgwụ
1. Deflazacort nwere potassium mmetụta pụrụ iche, yabụ a ga-eme nlekọta mgbe ejiri ya na njikọta na diuretics.
2. Mgbe ejiri ọgwụ ọjọọ jiri ọgwụ enzymatic (RIFAMPICIN, phenobarbital, wdg), glucocortoids kwesịrị ịmụba n'ụzọ kwesịrị ekwesị.
3. Erythromycin na Estrogen nwere ike igbochi metabolism nke ngwaahịa a na ihe ndị na-arụ ọrụ, na usoro onunu ogwu kwesiri ilelata ọnụ mgbe ejikọtara ọnụ. Ngwongwo kemịkal acetone-hexane kristal, na-agbaze 45-256.5 ℃. [α] d + 62.3 Celsius (c = 0,5, chloroform).

Ojiji
Ọgbọ nke atọ glucocortorip ndị nwere mgbochi mkpali, mgbochi nfụkasị, na ụba gloconeogesis. N'ihi na nke mbụ na nke abụọ na nke abụọ na nke abụọ, ọrịa na-egbu egbu, ọrịa anụ ahụ, ọrịa na-arịa ọrịa, ọrịa hediopathic, hediopathies, hediopaties, wdg.


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