Hexarelinbụ sịntetikpeptide nke na-eto eto hormone secretagogue (GHS)na ikeGHSR-1a agonist, mepụtara iji kpalientọhapụ nke homonụ nke uto endogenous (GH).. Ọ bụ nkeezinụlọ ghrelin mimeticma mejupụtara amino acid isii (hexapeptide), na-enye nkwụsi ike nke metabolic yana mmetụta mwepụta GH siri ike ma e jiri ya tụnyere analogs mbụ dị ka GHRP-6.
A na-amụ Hexarelin n'ọtụtụ ebe maka ngwa ya naendocrinology, imefusị ahụ ike, mmezi obi, na ọgwụgwọ ịka nká, n'ihi ike ya na-ebuli elu GH naIhe na-eto eto dị ka insulin 1 (IGF-1)ọkwa na-enweghị iwebata homonụ nke mpụga ozugbo.
Hexarelin na-ejikọta naOnye na-anabata ihe nzuzo nke homonụ na-eto eto (GHSR-1a)na pituitary na hypothalamus, na-eṅomi omume nkeghrelin-agụụ nke anụ ahụ na homonụ na-ahapụ GH.
Omume physiological isi:
Na-akpali mwepụta GH pulsatile
Na-abawanye ikesaIGF-1ọkwa
Na-akwalitemmetụta anabolic(Uto akwara, mgbake)
Na-akwadometabolism abụbanacell ọhụrụ
Nwere ike igosicardioprotectivenamgbochi apoptoticmmetụta
N'adịghị ka ụfọdụ peptides GHS ndị ọzọ, Hexarelin na-eme yaadịghị abawanye cortisol ma ọ bụ prolactin, na-enye profaịlụ endocrine dị ọcha.
Na-akwalitedabere ahu ukammepe
Na-akwalitemmezi anụ ahụ na ịmaliteghachi
Agụrụ akwụkwọ nasarcopenia, cachexia, na mgbake mgbe ịwachara ahụ gasịrị
Ọmụmụ ihe izizi gosiriarụ ọrụ obi ka mmamgbe myocardial merụrụ ahụ
Na-ebelatafibrosis obina enhancesMpekere ejepụ ventricular aka ekpe
Enwere ike iji naobi mgbawanaobi ịka nkáụdị
Na-abawanyelipolysisna-emeziwanyeinsulin uche
Na-akwadoọgwụgwọ mgbochi ịka nkásite na GH / IGF-1 mkpali axis
Nwere ike inye aka idobenjupụta ọkpụkpụ na ahụ ike nkwonkwo
Ịdị ọcha ≥ 99%
Emepụtara site naNgwakọta peptide siri ike (SPPS)
Ụkpụrụ GMP, obere endotoxin na ihe mgbaze
Ọbịbịa na-agbanwe agbanwe:R&D n'ọtụtụ azụmaahịa