nke
Aha | Paclitaxel |
Nọmba CAS | 33069-62-4 |
Usoro ihe omimi | C47H51NO14 |
Ibu molekụla | 853.92 |
Nọmba EINECS | 608-826-9 |
Ebe esi nri | 774.66°C(buru amụma) |
Njupụta | 0,200 |
Ọnọdụ nchekwa | E mechiri ya na nkụ, chekwaa na friza, 2-8 Celsius |
Ụdị | Ntụ ntụ |
Agba | Ọcha |
Nkwakọ ngwaahịa | Akpa PE+Aluminom akpa |
Paclitaxel HCL; Paclitaxel (crude eke); Paclitaxelx; N-BENZYL-BETA-PHENYLISOSERINE ESTER; PACLITAXEL, TAXUS BREVIFOLIA; PACLITAXEL, TAXUS SPECIES; PACLITAXOL; PACLITAXEL
Nkọwa
Paclitaxel bụ monomeric diterpenoid nke ewepụtara na ogbugbo nke ọgwụ Taxus sitere n'okike.Nchọgharị isotope gosiri na paclitaxel jikọtara ya na microtubules polymerized na ọ naghị emeghachi omume na tubulin dimers na-enweghị polymerized.Mgbe ekpughere mkpụrụ ndụ ahụ na paclitaxel, a ga-akwakọba ọnụ ọgụgụ buru ibu nke microtubules na sel.Mkpokọta nke microtubules ndị a na-egbochi ọrụ dị iche iche nke mkpụrụ ndụ, karịsịa nkewa sel na-akwụsị na oge mitotic ma gbochie nkewa nkịtị nke sel.Site na Ⅱ-Ⅲ nyocha ụlọ ọgwụ, paclitaxel dabara adaba maka ọrịa kansa ovarian na ọrịa ara ara, ma nweekwa mmetụta ọgwụgwọ ụfọdụ na ọrịa kansa akpa ume, ọrịa cancer colorectal, melanoma, isi na olu kansa, lymphoma na ụbụrụ ụbụrụ.
Ngosipụta
Ọ na-enwe mmetụta dị mma na ọgwụgwọ ọrịa cancer ovarian na platinum na ọrịa cancer ovarian ndị ọzọ na-emegharị ahụ na ọrịa ara ara.Ọrịa cancer, ọrịa kansa eriri afọ nke elu, obere cell na ọrịa cancer akpa ume na-abụghị obere cell nwere echiche dị mma.
Eji
Jiri 1: Broad-spectrum anti-tumor botanicals maka ovarian cancer, ara ara, wdg.
Jiri 2: sara mbara-dị iche iche mgbochi tumor botanicals maka ọgwụgwọ nke ovarian cancer, ara ara na ọrịa ndị ọzọ.
Jiri 3: ọgwụ mgbochi.Maka ọgwụgwọ ọrịa cancer ara metastatic na ọrịa cancer ovarian metastatic.Broad-spectrum anti-tumor botanicals maka ọgwụgwọ ọrịa cancer ovarian, ọrịa ara ara na ọrịa ndị ọzọ.
Jiri 4: Ọgwụ mgbochi tumor dị irè;na-ejikọta na mpaghara N-terminal nke β-tubulin, na-akwalite ndị mbụ microtubule kwụsiri ike, na-eguzogide depolymerization, na-egbochi nkewa cell nkịtị na ọnyà na G2 / M usoro nke cell okirikiri.
Jiri 5: ọgwụ mgbochi microtubule, na-egbochi nkwụsịtụ site n'ịkwalite tubulin polymerization, na-ejigide nkwụsi ike tubulin, na igbochi cell mitosis.