API ndị ahịa ọgwụ
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Fmoc-His-Aib-OH
Fmoc-His-Aib-OH bụ ngọngọ ụlọ dipeptide eji na peptide synthesis, na-ejikọta Fmoc-echebe histidine na Aib (α-aminoisobutyric acid). Aib na-ewebata conformational rigidity, na-eme ka ọ bara uru maka imepụta peptides helical na kwụsiri ike.
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Boc-His(Trt)-Aib-Glu(OtBu)-Gly-OH
Boc-His (Trt) -Aib-Glu (OtBu) - Gly-OH bụ mpempe tetrapeptide echedoro nke ejiri na njikọ peptide na mmepe ọgwụ. Ọ nwere otu arụrụ arụ echekwabara nke ọma maka ijikọ na njiri mara Aib (α-aminoisobutyric acid) iji kwalite nkwụsi ike helix na nkwụsi ike.
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Ste-γ-Glu-AEEA-AEEA-OSU
Ste-γ-Glu-AEEA-AEEA-OSU bụ molekul njikọ lipidated synthetic emebere maka nnyefe ọgwụ ezubere iche yana mgbochi-ọgwụ conjugates (ADCs). Ọ nwere ọdụ stearoyl (Ste) hydrophobic, γ-glutamyl ezubere iche motif, AEEA spacers maka mgbanwe, yana otu OSu (NHS ester) maka njikọta nke ọma.
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Fmoc-Ile-αMeLeu-Leu-OH
Fmoc-Ile-αMeLeu-Leu-OH bụ ngọngọ ihe eji echekwa ihe eji eme ihe na-egosi α-methylated leucine, nke a na-ejikarị eme ihe n'ichepụta ọgwụ peptide iji kwalite nkwụsi ike nke metabolic na nhọrọ nnabata.
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Dodecyl Phosphocholine (DPC)
Dodecyl Phosphocholine (DPC) bụ ihe nchacha zwitterionic sịntetị nke a na-ejikarị na nyocha protein membrane na usoro ihe omimi, ọkachasị na NMR spectroscopy na crystallography.
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Caspofungin maka ọrịa antifungal
Aha: Caspofungin
Nọmba CAS: 162808-62-0
Usoro ihe omimi: C52H88N10O15
Ibu ibu: 1093.31
Nọmba EINECS: 1806241-263-5
Ebe esi mmiri: 1408.1± 65.0 °C (buru amụma)
Njupụta: 1.36± 0.1 g/cm3 (buru amụma)
Ọnụọgụ acidity: (pKa) 9.86±0.26 (buru amụma)
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Daptomycin 103060-53-3 maka Ọrịa na-efe efe
Aha: Daptomycin
Nọmba CAS: 103060-53-3
Usoro ihe omimi: C72H101N17O26
Ibu ibu: 1620.67
Nọmba EINECS: 600-389-2
Ebe mgbaze: 202-204°C
Ebe esi mmiri: 2078.2± 65.0 °C (buru amụma)
Njupụta: 1.45± 0.1 g/cm3 (buru amụma)
Ebe ọkụ ọkụ: 87 ℃
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Micafungin maka antifungal na antiviral
Aha: Micafungin
Nọmba CAS: 235114-32-6
Usoro ihe omimi: C56H71N9O23S
Ibu ibu: 1270.28
Nọmba EINECS: 1806241-263-5
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Vancomycin bụ ọgwụ nje glycopeptide a na-eji eme ihe maka nje bacteria
Aha: Vancomycin
Nọmba CAS: 1404-90-6
Usoro ihe omimi: C66H75Cl2N9O24
Ibu ibu: 1449.25
Nọmba EINECS: 215-772-6
Njupụta: 1.2882 (atụmatụ siri ike)
Ntụgharị ntụgharị: 1.7350 (atụmatụ)
Ọnọdụ nchekwa: Akara akọrọ, 2-8°C
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Vardenafil Dihydrochloride na-agwọ ọrịa akwụrụ 224785-91-5
Nọmba CAS: 224785-91-5
Usoro ihe omimi: C23H32N6O4S
Arọ molikula: 488.6
Nọmba EINECS: 607-088-5
Ebe mgbaze: 230-235°C
Njupụta: 1.37
Ebe ọkụ ọkụ: 9 ℃
Ọnọdụ nchekwa: Akara ala kpọrọ nkụ, chekwaa na friza, n'okpuru -20 Celsius
Ọnụọgụ acidity: (pKa) 9.86±0.20 (buru amụma)
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Orlistat 96829-58-2 na-ebelata mmịkọ nke abụba Sietary, na-ebute mbelata ibu
Nọmba CAS: 96829-58-2
Usoro ihe omimi: C29H53NO5
Ibu ibu: 495.73
Nọmba EINECS: 639-755-1
Ntụgharị akọwapụtara: D20-32.0°(c=1inchloroform)
Ebe esi mmiri: 615.9±30.0°C (buru amụma)
Njupụta: 0.976±0.06g/cm3(buru amụma)
Ọnọdụ nchekwa: 2-8°C
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A na-eji RU-58841 mee ihe dị ka mgbochi ntutu isi na isi nkwọcha nke nwoke
Nọmba:CB51396657
Aha: RU 58841
Nọmba CAS: 154992-24-2
Usoro ihe omimi: C17H18F3N3O3
Ibu ibu: 369.34
Nọmba EINECS: 1592732-453-0
